CK2/ERK8-IN-1

Datasheet MSDS
Catalog Number
SCAS20780
Product Name
CK2/ERK8-IN-1
CAS Number
1085822-09-8
Molecular Formula
C11H9Br4N3O2
Molecular Weight
534.82
Storage
Powder: -20°C for 3 years In solvent: -80°C for 6 months
Description
CK2/ERK8-IN-1 is a dual inhibitor of casein kinase 2 (CK2) (Ki: 0.25 µM) and ERK8 (IC50s: 0.50 μM) with pro-apoptotic efficacy. CK2/ERK8-IN-1 also binds to PIM1, DYRK1A, and HIPK2 (Kis: 8.65 µM, 11.9 µM, and 15.25 µM).
Target
CK2 ERK8 PIM1 HIPK2 DYRK1A Apoptosis
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