Catalog Number
SAUR11832
Product Name
BI847325
CAS Number
1207293-36-4
Synonyms
BI 847325 , BI-847325 , BI 847325 BI-847325
Molecular Formula
C29H28N4O2
Molecular Weight
464.56
Purity
97.54%
Solubility
DMSO: 18 mg/mL (38.7 mM) Ethanol: 1 mg/mL (2.15 mM) Water: <1 mg/mL ( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage
Powder: -20°C for 3 years In solvent: -80°C for 6 months
Description
BI-847325 is a selective dual inhibitor of MEK and aurora kinases (AK) with IC50 values of 4 and 15 nM for human MEK2 and AK-C, respectively.
Target
Aurora A (Human), Aurora B (Xenopus laevis), Aurora C (Human), MEK1, MEK2
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