Canertinib

Datasheet MSDS
Catalog Number
SEGF10183
Product Name
Canertinib
CAS Number
267243-28-7
Synonyms
PD-183805, CI-1033, PD-183805, CI-1033
Molecular Formula
C24H25ClFN5O3
Molecular Weight
485.94
Purity
100.00%
Solubility
DMSO: 10mM ( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage
Powder: -20°C for 3 years In solvent: -80°C for 6 months
Description
Canertinib (CI-1033, PD183805) is a pan-ErbB inhibitor that acts on EGFR and ErbB2 with IC50 of 1.5 nM and 9.0 nM, respectively, but has no inhibitory activity against PDGFR, FGFR, InsR, PKC, and CDK1/2/4. Phase 3。
Target
EGFR, HER2/ErbB2
Inquiry

new products