Ketanserin

Datasheet MSDS
Catalog Number
S5HT15525
Product Name
Ketanserin
CAS Number
74050-98-9
Synonyms
R41468 , Ketanserinum , Ketanserin tartrate
Molecular Formula
C22H22FN3O3
Molecular Weight
395.43
Purity
99.73%
Solubility
DMSO: 10mM ( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage
Powder: -20°C for 3 years In solvent: -80°C for 6 months
Description
Ketanserin is a quinazoline derivative and serotonin (5-hydroxytryptamine, 5HT) receptor subtype 2 (5-HTR2) antagonist with potential antihypertensive and antiplatelet activities. Following administration, ketanserin binds to and inhibits the signaling mediated by 5-HTR2, which inhibits serotonin-dependent vasoconstriction and platelet activation.
Target
5-HT2A, 5-HT2C (Human), 5-HT2C (Rat)
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