Regorafénib N-oxyde (M2)

Catalog Number
A10157
Product Name
Regorafénib N-oxyde (M2)
Structure
Regorafénib N-oxyde (M2)
CAS Number
835621-11-9
Molecular Formula
C21H15ClF4N4O4
Molecular Weight
498.81
Purity
98.03%
Solubility
DMSO: 10 mM ( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage
Powder: -20°C for 3 years In solvent: -80°C for 6 months
Description
Regorafénib N-oxyde M2 is an active metabolite of Regorafenib. Regorafenib is a multi-target inhibitor for VEGFR1/2/3, PDGFRβ, RET, Kit, and Raf-1 (IC50s: 13/4.2/46, 1.5, 22, 7, and 2.5 nM).
Target
Others
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