CEP-28122 mesylate salt (1022958-60-6 free base)

Datasheet MSDS
Catalog Number
SALK10038
Product Name
CEP-28122 mesylate salt (1022958-60-6 free base)
Synonyms
CEP-28122 mesylate salt (1022958-60-6 free base)
Molecular Formula
C29H39ClN6O6S
Molecular Weight
635.17
Purity
99.19%
Solubility
DMSO: 6.4 mg/mL (10.08 mM) ( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage
Powder: -20°C for 3 years In solvent: -80°C for 6 months
Description
CEP-28122 mesylate salt, a diaminopyrimidine derivative, is a potent, selective, and orally bioavailable ALK inhibitor, with an IC50 value of 1.9 nM for recombinant ALK kinase activity. CEP-28122 has antitumor activity in experimental models of ALK-positive human cancers. CEP-28122 mesylate salt has good pharmacodynamic and pharmacokinetic activity.
Target
Others
Inquiry

new products